Buy Ciclazindol (anorectic) Cas 37751-39-6
Buy Ciclazindol (anorectic) Cas 37751-39-6
Buy Ciclazindol (anorectic) Cas 37751-39-6
Ciclazindol (WY-23409) is an antidepressant and anorectic[2] drug of the tetracyclic[citation needed] chemical class that was developed in the mid to late 1970s, but was never marketed.[3][4] It acts as a norepinephrine reuptake inhibitor, and to a lesser extent as a dopamine reuptake inhibitor.[3][5] Ciclazindol has no effects on the SERT, 5-HT receptors, mACh receptors, or α-adrenergic receptors, and has only weak affinity for the H1 receptor.[5][6][7] As suggested by its local anesthetic properties,[6] ciclazindol may also inhibit sodium channels. It is known to block potassium channels as well.[8][9]
The dosage in human volunteers is stated to be 25 mg daily.[1] However, doses of up to 200 mg have also been reported.[2] This is surprising since the dosage of mazindol is only 2-4 mg per day.
Ciclazindol is reported to have an IC50 of 1.3 nM for the dopamine transporter (cmp 23).[10]
See also
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Ciclazindol 37751-39-6 | MedChemExpress
MedChemExpress provides Ciclazindol CAS 37751-39-6, related Reference Standards, Isotope-Labeled or GMP Grade Compounds, …
Ciclazindol
Synonym(s): WY-23409
- CAS No.:37751-39-6
- Formula:C17H15ClN2O
- Molecular Weight:298.77
IUPAC Name: 10-(3-chlorophenyl)-2,3,4,10-tetrahydropyrimido[1,2-a]indol-10-ol
InChIKey: VKQDZNZTPGLGFD-UHFFFAOYSA-N
SMILES: OC1(C2=CC(Cl)=CC=C2)C3=C(C=CC=C3)N4C1=NCCC4
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Ciclazindol | 37751-39-6 – ChemicalBook
Ciclazindol (CAS 37751-39-6) information, including chemical properties, structure, melting point, boiling point, …
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Ciclazindol (WY-23409) | Antidepressant | MedChemExpress
Ciclazindol (WY-23409) is an orally active antidepressant. Ciclazindol can inhibit the reuptake of norepinephrine. Ciclazindol also …
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CAS No.: 37751-39-6
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Molecular Weight: 298.77
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Formula: C 17 H 15 ClN 2 O
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Ciclazindol | 37751-39-6, Ciclazindol Formula – ECHEMI
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Ciclazindol (free base) | CAS#37751-39-6 (free base) | inhibitor | MedKoo
Ciclazindol (free base) is a noradrenaline uptake inhibitor. This product is currently not in stock but may be available through custom …
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